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Letovišče Habubu jesen dp dr kappa antagonist Aditiv Vzdihanje Vernik

Nalfurafine, a G-Protein–Biased KOR (Kappa Opioid Receptor) Agonist, Enhances the Diuretic Response and Limits Electrolyte Losses to Standard-of-Care Diuretics | Hypertension
Nalfurafine, a G-Protein–Biased KOR (Kappa Opioid Receptor) Agonist, Enhances the Diuretic Response and Limits Electrolyte Losses to Standard-of-Care Diuretics | Hypertension

Discovery of Small Molecule Kappa Opioid Receptor Agonist and Antagonist Chemotypes through a HTS and Hit Refinement Strategy | ACS Chemical Neuroscience
Discovery of Small Molecule Kappa Opioid Receptor Agonist and Antagonist Chemotypes through a HTS and Hit Refinement Strategy | ACS Chemical Neuroscience

Proteomes | Free Full-Text | Exploring Morphine-Triggered PKC-Targets and Their Interaction with Signaling Pathways Leading to Pain via TrkA
Proteomes | Free Full-Text | Exploring Morphine-Triggered PKC-Targets and Their Interaction with Signaling Pathways Leading to Pain via TrkA

Anti-HLA DR + DP + DQ antibody [CR3/43] (ab7856) | Abcam
Anti-HLA DR + DP + DQ antibody [CR3/43] (ab7856) | Abcam

Pharmaceuticals | Free Full-Text | In Vitro, In Vivo and In Silico Characterization of a Novel Kappa-Opioid Receptor Antagonist
Pharmaceuticals | Free Full-Text | In Vitro, In Vivo and In Silico Characterization of a Novel Kappa-Opioid Receptor Antagonist

I'll Be Back”: The Resurrection of Dezocine | ACS Medicinal Chemistry Letters
I'll Be Back”: The Resurrection of Dezocine | ACS Medicinal Chemistry Letters

Putative interaction modes of morphine-based high-affinity... | Download Scientific Diagram
Putative interaction modes of morphine-based high-affinity... | Download Scientific Diagram

Preventing Morphine-Seeking Behavior through the Re-Engineering of Vincamine's Biological Activity | Journal of Medicinal Chemistry
Preventing Morphine-Seeking Behavior through the Re-Engineering of Vincamine's Biological Activity | Journal of Medicinal Chemistry

6,5‐Fused Ring, C2‐Salvinorin Ester, Dual Kappa and Mu Opioid Receptor Agonists as Analgesics Devoid of Anxiogenic Effects** - Akins - 2022 - ChemMedChem - Wiley Online Library
6,5‐Fused Ring, C2‐Salvinorin Ester, Dual Kappa and Mu Opioid Receptor Agonists as Analgesics Devoid of Anxiogenic Effects** - Akins - 2022 - ChemMedChem - Wiley Online Library

Frontiers | Opioid Receptor-Mediated Regulation of Neurotransmission in the Brain
Frontiers | Opioid Receptor-Mediated Regulation of Neurotransmission in the Brain

Molecules | Free Full-Text | Mechanistic Characterization of the Pharmacological Profile of HS-731, a Peripherally Acting Opioid Analgesic, at the µ-, δ-, κ-Opioid and Nociceptin Receptors
Molecules | Free Full-Text | Mechanistic Characterization of the Pharmacological Profile of HS-731, a Peripherally Acting Opioid Analgesic, at the µ-, δ-, κ-Opioid and Nociceptin Receptors

Dynamic lateral organization of opioid receptors (kappa, muwt and muN40D) in the plasma membrane at the nanoscale level - Rogacki - 2018 - Traffic - Wiley Online Library
Dynamic lateral organization of opioid receptors (kappa, muwt and muN40D) in the plasma membrane at the nanoscale level - Rogacki - 2018 - Traffic - Wiley Online Library

Prefrontal Cortical Kappa-Opioid Receptor Modulation of Local Neurotransmission and Conditioned Place Aversion | Neuropsychopharmacology
Prefrontal Cortical Kappa-Opioid Receptor Modulation of Local Neurotransmission and Conditioned Place Aversion | Neuropsychopharmacology

Frontiers | The role of endogenous opioid neuropeptides in neurostimulation-driven analgesia
Frontiers | The role of endogenous opioid neuropeptides in neurostimulation-driven analgesia

Structural Assessment of Agonist Efficacy in the μ-Opioid Receptor: Morphine and Fentanyl Elicit Different Activation Patterns | Journal of Chemical Information and Modeling
Structural Assessment of Agonist Efficacy in the μ-Opioid Receptor: Morphine and Fentanyl Elicit Different Activation Patterns | Journal of Chemical Information and Modeling

Antagonists of the kappa opioid receptor - ScienceDirect
Antagonists of the kappa opioid receptor - ScienceDirect

Discovery of Small Molecule Kappa Opioid Receptor Agonist and Antagonist Chemotypes through a HTS and Hit Refinement Strategy | ACS Chemical Neuroscience
Discovery of Small Molecule Kappa Opioid Receptor Agonist and Antagonist Chemotypes through a HTS and Hit Refinement Strategy | ACS Chemical Neuroscience

Early life stress dysregulates kappa opioid receptor signaling within the lateral habenula - ScienceDirect
Early life stress dysregulates kappa opioid receptor signaling within the lateral habenula - ScienceDirect

The Role of Dynorphin and the Kappa Opioid Receptor in the Symptomatology of Schizophrenia: A Review of the Evidence
The Role of Dynorphin and the Kappa Opioid Receptor in the Symptomatology of Schizophrenia: A Review of the Evidence

Pharmaceuticals | Free Full-Text | Druggable Targets and Compounds with Both Antinociceptive and Antipruritic Effects
Pharmaceuticals | Free Full-Text | Druggable Targets and Compounds with Both Antinociceptive and Antipruritic Effects

Lion's Mane contains kappa agonist - Supplements - LONGECITY
Lion's Mane contains kappa agonist - Supplements - LONGECITY

Synthesis and Structure–Activity Relationships of 5′-Aryl-14-alkoxypyridomorphinans: Identification of a μ Opioid Receptor Agonist/δ Opioid Receptor Antagonist Ligand with Systemic Antinociceptive Activity and Diminished Opioid Side Effects | Journal ...
Synthesis and Structure–Activity Relationships of 5′-Aryl-14-alkoxypyridomorphinans: Identification of a μ Opioid Receptor Agonist/δ Opioid Receptor Antagonist Ligand with Systemic Antinociceptive Activity and Diminished Opioid Side Effects | Journal ...

Role of RGS12 in the differential regulation of kappa opioid receptor-dependent signaling and behavior | Neuropsychopharmacology
Role of RGS12 in the differential regulation of kappa opioid receptor-dependent signaling and behavior | Neuropsychopharmacology

Kappa Opioid Receptor Activation Potentiates the Cocaine-Induced Increase in Evoked Dopamine Release Recorded In Vivo in the Mouse Nucleus Accumbens | Neuropsychopharmacology
Kappa Opioid Receptor Activation Potentiates the Cocaine-Induced Increase in Evoked Dopamine Release Recorded In Vivo in the Mouse Nucleus Accumbens | Neuropsychopharmacology

Frontiers | Crosstalk Between Kappa Opioid and Dopamine Systems in Compulsive Behaviors
Frontiers | Crosstalk Between Kappa Opioid and Dopamine Systems in Compulsive Behaviors